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Pri zdravih osebah, ki so med klinično študijo 7 dni sočasno prejemale ritonavir v obliki 100 mg kapsul dvakrat dnevno in flutikazonpropionat v odmerku 50 µg intranazalno(4- krat dnevno) so ugotovili, da so se vrednosti flutikazonpropionata v plazmi znatno povečale, intrinzične vrednosti kortizola pa zmanjšale za približno 86%(90% interval zaupanja; 82- 89%.
Fluticasone propionate(interaction with ritonavir): in a clinical study where ritonavir 100 mg capsules bid were co-administered with 50 µg intranasal fluticasone propionate(4 times daily) for 7 days in healthy subjects, the fluticasone propionate plasma levels increased significantly, whereas the intrinsic cortisol levels decreased by approximately 86%(90% confidence interval 82-89%.
Flutikazonpropionat(interakcija z ritonavirjem): pri zdravih osebah, ki so med klinično študijo 7 dni sočasno prejemale ritonavir v obliki 100 mg kapsul dvakrat dnevno in flutikazonpropionat v odmerku 50 µg intranazalno(4- krat dnevno), so ugotovili, da so se vrednosti flutikazonpropionata v plazmi znatno povečale, intrinzične vrednosti kortizola pa zmanjšale za približno 86%(90% interval zaupanja; 82- 89%.
Fluticasone propionate(interaction with ritonavir): in a clinical study where ritonavir 100 mg capsules twice daily were co- administered with 50 μ g intranasal fluticasone propionate(4 times daily) for seven days in healthy subjects, the fluticasone propionate plasma levels increased significantly, whereas the intrinsic cortisol levels decreased by approximately 86%(90% confidence interval 82- 89%.
Ledvični očistek flutikazonpropionata je zanemarljiv.
The renal clearance of fluticasone propionate is negligible.
Izločanje Ledvični očistek flutikazonpropionata je zanemarljiv.
The renal clearance of fluticasone propionate is negligible.
Ena inhalacija 50 mikrogramov salmeterola in 500 mikrogramov flutikazonpropionata dvakrat na dan.
One inhalation of 50 micrograms salmeterol and 500 micrograms fluticasone propionate twice daily.
Flutikazonpropionata je mogoče.
When fluticasone propionate is inhaled.
Nekatera od teh zdravil lahko povečajo količino salmeterola ali flutikazonpropionata v telesu.
Some of these medicines may increase the amount of salmeterol or fluticasone propionate in your body.
Nekatera od teh zdravil lahko povečajo količino salmeterola ali flutikazonpropionata v telesu.
Some of these medicines may increase the amount of fluticasone propionate or salmeterol in your body.
in 500 mikrogramov flutikazonpropionata.
500 micrograms of fluticasone propionate.
Zdravilo Aerivio Spiromax ni primerno za zdravljenje astme, če je fiksna kombinacija odmerka salmeterola in flutikazonpropionata potrebna prvič.
Aerivio Spiromax is not intended as the treatment of asthma when a fixed-dose combination of salmeterol and fluticasone propionate is required for the first time.
tem medsebojnem delovanju ni, a pričakovati je mogoče izrazito povečanje koncentracije flutikazonpropionata v plazmi.
for inhaled fluticasone propionate, but a marked increase in fluticasone propionate plasma levels is expected.
in 465 mikrogramov flutikazonpropionata.
500 micrograms fluticasone propionate.
Plazemske vrednosti flutikazonpropionata so se znatno povečale,
The fluticasone propionate plasma levels increased significantly,
Absolutna biološka uporabnost inhaliranega flutikazonpropionata pri zdravih preiskovancih je med približno 5 in 11% nominalnega odmerka, odvisno od uporabljene inhalacijske naprave.
The absolute bioavailability of a single dose of inhaled fluticasone propionate in healthy subjects varies between approximately 5 to 11% of the nominal dose depending on the inhalation device used.
V primeru odsotnosti enega ali dveh kriterijev za ocenitev stopnje bolezni očitna korist pri začetnem vzdrževalnem zdravljenju, v primerjavi z uporabo inhalacijskega flutikazonpropionata samega, ni bila dokazana.
A clear benefit has not been shown as compared with inhaled fluticasone propionate alone used as initial maintenance therapy when one or two of the criteria of severity are missing.
Za razporeditev flutikazonpropionata so značilni velik očistek iz plazme(1.150 ml/min),
The disposition of fluticasone propionate is characterised by high plasma clearance(1150 mL/min),
S študijami na živalih z ločenim dajanjem salmeterola in flutikazonpropionata so ugotovili, da edino skrb glede varnosti uporabe pri ljudeh predstavljajo učinki, povezani s pretiranim farmakološkim delovanjem.
The only safety concerns for human use derived from animal studies of salmeterol and fluticasone propionate given separately were effects associated with exaggerated pharmacological actions.
Sočasna uporaba zdravila EVOTAZ in flutikazonpropionata ali drugih inhalacijskih ali nazalnih kortikosteroidov ni priporočljiva,
Concomitant use of EVOTAZ and fluticasone propionate or other inhaled or nasal corticosteroids is
za kar je potreben prehod na drugo fiksno kombinacijo odmerka salmeterola in flutikazonpropionata, ki vsebuje manjši odmerek inhalacijskega kortikosteroida.
therefore a change to an alternative fixed-dose combination of salmeterol and fluticasone propionate containing a lower dose of the inhaled corticosteroid is required.
so bile izvedene z enako fiksno kombinacijo odmerkov salmeterolijevega ksinafoata in flutikazonpropionata, vendar s predhodno odobrenim zdravilom;
were carried out with this same fixed-dose combination, salmeterol xinafoate and fluticasone propionate, but studied a previously authorised product;